◆ Synthesis: Synthesis of Enantiopure Quaternary Prolines by a Metathesis Process of 2,5-Ethenoproline Derivatives

Javier Carreras, Alberto Avenoza, Jesús H. Busto, and Jesús M. Peregrina

A novel azabicyclic amino acid was synthesized in both enantiopure forms. The ring-opening metathesis of methyl N-(tert-butoxycarbonyl)-7-azabicyclo[2.2.1]hept-2-ene-1-carboxylates was used as a method for accessing a new family of enantiopure proline analogues.


Synthesis 2010, 19, 3353; doi: 10.1055/s-0030-1257907